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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T69537 | Difelikefalin HCl | ||
Difelikefalin HCl is a κ-opioid receptor (KOR) agonist. It activates KOR in HEK293 cells expressing the human receptor (EC50 = 0.16 nM in a transactivation assay) and inhibits forskolin-induced cAMP production in R1.G1 m... | |||
TP2485 | difelikefalin acetate(1024828-77-0 Free base) | Opioid Receptor | |
is a ketone and a building block. | |||
TP2501 | Difelikefalin acetate | Difelikefalin acetate(1024828-77-0 free base),CR 845 acetate,FE 202845 acetate | Opioid Receptor |
Difelikefalin acetate (CR 845 acetate) is a peripherally restricted kappa opioid receptor agonist. CR845 exhibit low P450 CYP inhibition and low penetration into the brain. |